![Ni antipsychotic gani ni anticholinergic? Ni antipsychotic gani ni anticholinergic?](https://i.answers-medical.com/preview/medical-health/13939095-which-antipsychotics-are-anticholinergic-j.webp)
Video: Ni antipsychotic gani ni anticholinergic?
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2024 Mwandishi: Michael Samuels | [email protected]. Mwisho uliobadilishwa: 2023-12-16 01:52
FGAs zenye nguvu ndogo na clozapine zina uwezekano mkubwa wa kusababisha athari ya anticholinergic ; olanzapine na quetiapine zimeonyeshwa kufanya hivyo kwa kipimo kikubwa.
Kwa hivyo, je, quetiapine ni kinzacholinergic?
Hii inamaanisha quetiapini ni dopamine, serotonini, na adrenergic antagonist, na antihistamine yenye nguvu na zingine anticholinergiki mali. Quetiapine hufunga sana kwa vipokezi vya serotonini; dawa hufanya kama agonist sehemu katika 5-HT1A vipokezi.
Baadaye, swali ni, ni antipsychotic gani ambayo ina uwezekano mdogo wa kusababisha dyskinesia ya kuchelewa? Risperidone , olanzapine , quetiapini , na clozapine kuwa na hatari ndogo ya dyskinesia ya kuchelewa.
Pia Jua, je olanzapine ni dawa ya anticholinergic?
Mfano wa anticholinergic shughuli ya antipsychotic ya atypical dawa . HALI YA ASILI: Dawa za kuzuia magonjwa ya akili clozapine , olanzapine , na quetiapine zina ushirika mkubwa kwa vipokezi vya muscarinic katika vitro, wakati aripiprazole, risperidone , na ziprasidone hawana.
Je! SSRI ipi ina athari ya anticholinergic zaidi?
The vizuizi vya kuchukua tena serotonini (SSRIs), kama citalopram (Celexa ) na duloxetini (Cymbalta), hutumiwa kwa kawaida kutibu unyogovu kwa watu wa rika zote. Baadhi yao wana athari kali za kinzakolinajiki kuliko wengine, lakini zaidi ya yote wana athari ya chini ya kinzakolinajiki.
Ilipendekeza:
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Sababu. Dalili za Extrapyramidal husababishwa sana na dawa za kawaida za kuzuia magonjwa ya akili ambazo hupinga receptors za D2. Dawa za kawaida za kuzuia magonjwa ya akili zinazohusiana na EPS ni haloperidol na fluphenazine
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Mifano ya phenothiazine antipsychotic ni: prochlorperazine (Compazine, Compro, Procomp), chlorpromazine (Promapar, Thorazine), fluphenazine (Permitil, Prolixin), perphenazine, trifluoperazine (Stelazine), thioridazine (Mellaril), na. mesoridazine (haipatikani tena nchini Merika)
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Utaratibu uliowekwa wa shughuli za kifafa kutokana na kundi hili la dawa unaweza kuhusishwa na ongezeko la kutolewa kwa katekisimu na kusababisha msisimko wa kusisimua. Kutolewa kwa catecholamine kupita kiasi kunaweza kukomesha kifafa kupitia kupoteza usingizi na mafadhaiko ya mwili. Dawa zote za kuzuia magonjwa ya akili zinaweza kupunguza kizingiti cha mshtuko
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Dawa za cholinergic huongeza athari za acetylcholine, na kuongeza vitendo vya mfumo wa neva wa parasympathetic. Dawa za anticholinergic huzuia athari za asetilikolini, kupunguza vitendo vya parasympathetic na kuongeza huruma. Dawa za cholinergic hutumiwa kutibu glaucoma na myasthenia gravis
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Phenelzine (Nardil, Nardelzine) ni kizuizi kisichochagua na kisichoweza kutenduliwa cha monoamine oxidase (MAOI) cha darasa la hydrazine ambacho hutumika kama kizuia mfadhaiko na wasiwasi